赵金浩 教授,博导

发布时间:2024-04-06浏览次数:7142


 赵金浩 教授, 博士生导师,


浙江大学农学院植保系,农药与环境毒理研究所

地址:杭州市余杭塘路866号,浙江大学紫金港校区-西区农科教大楼A511

邮编:310029

电话:0571-87075689

传真:0571-87075689

Emailjinhaozhao@zju.edu.cn



更多信息请见浙江大学教师个人主页:https://person.zju.edu.cn/jhzhao


研究方向

· 农药缓控释材料/纳米-缓控释制剂

· 农药靶向递送及剂量传递

· 基于天敌引诱的绿色防控

· 农药化学生物学及应用化学

 

个人简介

赵金浩,教授,博士生导师,有机化学专业博士,药学博士后,浙江东阳人。先后主持国家自然科学基金3项、国家科技支撑重大专项1项、国家科技计划十二五、十三五、十四五重点研发项目子课题5项、浙江省科技厅重大专项1项、科技厅面上项目2项,以及企业委托清洁生产工艺项目。近几年在Acs NanoSmallChem. Eng. J. J. Hazard Mat.J. Agric. Food Chem等国内外期刊发表相关SCI文章80多篇,授权中国发明专利30件,美国专利1, 其中专利成果转4。部分研究成果曾获得中国石化协会科技进步一等奖3项、浙江省科技进步一等奖2项。2009.9获得浙江大学青年骨干教师赴国外高水平大学合作研究计划经费资助,赴美国密西根大学生命科学学院学习年,访问交流学者。2011年入选浙江省151人才工程第三层次培养人员。已培养博、硕士生近40多名。

 

科研项目

纵向(主持):

15. 国家自然科学基金面上项目,项目编号:323725752024.01-2027.12

14.“十四五国家重点研发计划农药农机农艺三融合省力化精准施药技术与产业化项目,子课题,2023.12-2027.12

13.“十四五国家重点研发计划农药靶向传输释放调控与协同控害技术创新与应用子课题,2022.11-2026.

12. 国家自然科学基金面上项目,项目编号:318720222019.01-202022.12.
11.“十三五国家重点研发项目北方玉米化肥农药减施技术集成研究与示范子课题, 2017.1-2020.12
10.“十三五国家重点研发计划项目子课题,项目编号:SQ2017ZY0600592017.1-2020.12

9. 国家自然科学基金青年基金,项目编号:307005322008.12010.12

8. 浙江省科技厅重大专项重点项目,2008.6-2011.5

7. 国家科技重大专项课题-重大新药创制,2009.01-2010.12

6国家科技支撑计划课题,子项目,2011.1-2015.3.

5省科技厅面上项目:新颖高效杀螨剂螺螨酯的研制及产业化技术开发,30万,2008.1-2010.12

4浙江省科技厅公益面上项目:外来入侵红火蚁化学信息素的合成及其诱捕防治技术研究,2015.01.01-2016.12.31

3浙江大学基本科研业务费专项资金-青年科研创新专项项目;2012.3-2013.12

2农业部项目:农药残留代谢研究制定中比例推算研究. 2012.10.20-2012.12.31

1. 教育厅一般项目,2011.10.1-2013.10.31

 

横向(主持)

4. 企业委托重大横向项目:YX连续化工艺流程开发与生产转化,2021.12-2026.12

3. 企业委托重大横向项目:YX新工艺技术生产转化, 2020.06.01  - 2024.12.31

2.企业委托横向项目:BYTKLT的制备工艺与优化2020.06.01  -- 2020.12.31 

1. 企业委托重大横向项目:LSYX工艺开发和添加剂配方研究,2017.12.1-2020.11.30

  等等.....

转让专利:

1转让中国发明专利2项, 专利权转让,2020.11

2转让中国发明专利1项,专利独占许可实施三年,2020.11.16-2023.11.15

3转让中国发明专利1项,专利独占许可实施六年,2014.12.16-020.12.15

 

已发表SCI论文:

2024

85. Bin Yu, Jingli Cheng, Yun Fang, Zhengang Xie, Qiuyu Xiong, Haonan Zhang, Wenxuan Shang, Frederik R. Wurm, Wenlong Liang*, Fanglin Wei*, and Jinhao Zhao*. Multi-Stimuli-Responsive, Topology-Regulated, and Lignin-Based Nano/Microcapsules from Pickering Emulsion Templates for Bidirectional Delivery of Pesticides.  ACS Nano, 2024, 18:10031-10044. 

84. Yun Fang, Zhengang Xie, Haonan Zhang, Qiuyu Xiong, Bin Yu, Jingli ChengWenxuan Shang, Jinhao Zhao*. Near-infrared-responsive CuS@Cu-MOF nanocomposite with high foliar retention and extended persistence for controlling strawberry anthracnose.Journal of Controlled Release,  2024(367): 837-847.

2023

83Wenxuan Shang, Qiuyu Xiong, Zhengang Xie , Jingli Cheng, Bin Yu, Haonan Zhang, Yehua Su* & Jinhao Zhao*. Functional, ecofriendly, and starchbased nanocarriers with sustained release of carvacrol for persistent control of tomato gray moldCrop Health2023(1):13. 

82. Qiuyu Xiong, Wenlong Liang, Wenxuan Shang, Zhengang Xie, Jingli Cheng, Bin Yu, Yun Fang, Li Sun, and Jinhao Zhao*. Bidirectional Uptake, Transfer, and Transport of Dextran-based Nanoparticles in Plants for Multidimensional Enhancement of Pesticide Utilization. Small 2023, 2305693.

81. Jingli Cheng, Haonan Zhang , Bin Yu , Qiuyu Xiong, Zhengang Xie , Qi Zhang , Rong Wang , Yehua Su , Jinhao Zhao*. Recyclable bispyridine functionalized polyacrylonitrile fibers as ligand of Cu(II) for A3 coupling reaction. Reactive and Functional Polymers, 2023 (193):105767.

80. Zhengang Xie, Qiuyu Xiong, Yun Fang, Qi Zhang, Wenlong Liang, Jingli Cheng, Wenxuan Shang, Wei Zhao, and Jinhao Zhao*. Novel Biodegradable Composite Mulch Film Embedded with Temperature-Responsive Pesticide Microcapsules for Durable Control of Phytophthora Root Rot on Soybean. ACS Sustainable Chemistry Engineering2023,11:9868-9879

 79. Haonan Zhang , Wenlong Liang , Jian Xiao*, Jinhao Zhao*. Functional fiber with bis (N-heterocyclic carbene) structure prevents Pd(0) nanoparticle agglomeration for an efficient and recyclable Heck reaction. Chemical Engineering Journal. 2023, (455) :140592 (IF5 =15.10)

2022

78. Wenlong Liang, Jingli Cheng, Jiadong Zhang, Qiuyu Xiong, Maojun Jin*, Jinhao Zhao*pH-Responsive On-Demand Alkaloids Release from Core–Shell ZnO@ZIF-8 Nanosphere for Synergistic Control of Bacterial Wilt Disease. ACS Nano, 2022, 16,2762-2773  (IF5 =17.09)

77. Zhengang Xie1, Wenlong Liang1, Qiuyu Xiong, Yanyan Zhao, Jingli Cheng, Xianbin Li*, Jinhao Zhao*, Acetalated dextran microparticles for the smart delivery of pyraclostrobin to control Sclerotinia diseases. Carbohydrate Polymers, 2022291, 119576.  

76. Wenlong Liang1, Jiadong Zhang1, Frederik R. Wurm, Rong Wang, Jingli ChengZhengang Xie, Xianbin Li *, Jinhao Zhao* Lignin-based non-crosslinked nanocarriers: A promising delivery system of pesticide for development of sustainable agriculture . International Journal of Biological Macromolecules. 2022220472–481

75. Jinhao Zhao, Minmin Liang, Zhongyan Wang, Yanyan 75. Zhao, Jingli Cheng*,  Yongjun Du*. Evaluation and optimization of blends for attracting Trichogramma dendrolimi based on semiochemicals mediating tritrophic interactions in the orchard habitat. Biological Control, 2022, 173: 104998

74. Hui-Liang Hua, Guo-Ping Wang, Jing-Li Cheng, Yong-Min, Liang,* and Jin-Hao Zhao*. H2O2-Promoted Alkoxyalkylation of Terminal Alkynes Employing Two Strategies with Transition-Metal-Free Conditions, Asian J. org. chem. 2022,11, e202100726.

2021

73. Wenlong Liang, Zhengang Xie, Jingli Cheng, Douxin Xiao, Qiuyu Xiong, Qiangwei Wang, Jinhao Zhao*, Wenjun Gui*. A Light-Triggered pH-Responsive Metal−Organic Framework for Smart Delivery of Fungicide to Control Sclerotinia Diseases of Oilseed Rape. ACS Nano2021, 15, 6987-6997.  (IF5 =17.09)

72. Douxin Xiao, Jingli Cheng, Wenlong Liang, Lianli Sun,*, Jinhao Zhao,* .Metal-phenolic coated and prochloraz-loaded calcium carbonate carriers with pH responsiveness for environmentally-safe fungicide deliveryChemical Engineering Journal2021, (418) :129274. (IF5 =15.10)

71. Wenlong Liang, Biao Wang, Jingli Cheng, Douxin Xiao, Zhengang Xie, Jinhao Zhao*. 3D, Eco-friendly Metal-organic Frameworks@Carbon Nanotube Aerogels Composite Materials for Removal of Pesticides in Water. Journal of Hazardous Materials. 2021401: 123718. (IF5=13.60) 

70. Douxin Xiao , Wenlong Liang , Zhengang Xie , Jingli Cheng , Yongjun Du , Jinhao Zhao * . A temperature-responsive release cellulose-based microcapsule loaded with chlorpyrifos for sustainable pest control. Journal of Hazardous Materials. 2021403: 123654 (IF5=13.60)

2020

69. Yirong Guo1 , Rubing Zou1, Fangfang Sia, Wenlong Liang , Tianyi Zhang , Yunyun Chang , Xvsheng Qiao , Jinhao Zhao*. A sensitive immunoassay based on fluorescence resonance energy transfer from up-converting nanoparticles and graphene oxide for one-step detection of imidacloprid. Food Chemistry. 2020. 2021,335:127609

68. Jinhao zhao, Zhongyan Wang, Zhongshan Li, Jiayu Shi, Ling Meng, Guorong Wang, Jingli Cheng, Yongjun Du*. Development of lady beetle attractants from floral volatiles and other semiochemicals for the biological control of aphids. Journal of Asia-Pacific Entomology. 2020, 23: 1023-1029.

67.  She, S., Zhao, Y., Kang, B., Chen, C., Chen, X., Zhang, X., ... & Zhao, Jinhao. Combined inhibition of JAK1/2 and DNMT1 by newly identified small-molecule compounds synergistically suppresses the survival and proliferation of cervical cancer cells. Cell Death & Disease, 2020, 11(9), 1-16. (IF5= 9.00)

66. Li, Anbang Li, Zhongshan Zhao,Yang Yao,Tingting Cheng, Jingli, Zhao, Jinhao*. Design, Synthesis, and Antifungal Activity of Novel Pyrazole-Thiophene Carboxamide. Chinese Journal of Organic Chemistry, 2020, 40: 2836~2844.

65. ZHAO Yang, CHENG Jingli* , XIE Zhengang, FANG Shaowei and ZHAO Jinhao *. Syntheses and Insecticidal Activity of Spirocyclic Tetronic Acid Derivatives Containing Oxime Ether Moiety.Chemical Research in Chinese Universities. 2020 , 36(5): 810-815

64. Biao Wang, Yong Yang1 , Yu Lu , Wei Wang , Qiangwei Wang , Xiaowu Dong , Jinhao Zhao*.  Rapid and efficient removal of acetochlor from environmental water using Cr-MIL-101 sorbent modified with 3, 5-Bis(trifluoromethyl) phenyl isocyanate. Science of the Total Environment, 2020, 710: 135512

63.  程敬丽,肖豆鑫,梁文龙,方逊,张家栋,赵金浩*. pH 响应性吡唑醚菌酯/沸石咪唑酯骨架材料纳米颗粒的制备及抑菌活性农药学学报2022, 24(1): 105-113(封面论文).

62. 敬丽,梁文龙,张家栋,熊秋雨,赵金浩*. 基于粒径和形貌视角下探究微乳剂是否为纳米农药浙江农业科学2022, 63(11): 2636-2639.

61.  程敬丽张家栋,梁敏敏,肖豆鑫,赵金浩吡丙醚乙基纤维素微胶囊的制备及其性能研究,农药2021,  60(12): 882-886

60. 程敬丽,李安邦,肖豆鑫,赵金浩*. N-取代苯基-4-(1-甲基-1H-吡唑-5-)噻吩-2-甲酰胺的合成、杀菌活性及分子对接农药学学报2021, 23(5): 877-885.

59. 王忠燕,李中珊,董环,程敬丽,杜永均,赵金浩*. 基于智能测报的沈阳亚洲玉米螟监测浙江农业科学2020, 1: 101-103

2019

58. Douxin Xiao,§  Wenlong Liang, § Zhongshan Li, Jingli Cheng, Yongjun Du, Jinhao Zhao*. High Foliar Affinity Cellulose for the Preparation of Efficient and Safe Fipronil Formulation.Journal of Hazardous Materials. 2019.121408. 

57. Wenlong Liang, Yang Zhao, Douxin Xiao, Jingli Cheng, Jinhao Zhao* . A biodegradable water-triggered chitosan/hydroxypropyl methylcellulose pesticide mulch film for sustained control of Phytophthora sojae in soybean (Glycine max L. Merr.). Journal of Cleaner Production. 2019. 245: 118943.

56. Douxin Xiao, Jingli Cheng, Wenlong Liang, Cheng Cheng, Qiangwei Wang, Rongyao Chai, Zhenlong Yan, Yongjun Du, and Jinhao Zhao*. Innovative Approach to Nano Thiazole-Zn with Promising Physicochemical and Bioactive Properties by Nanoreactor Construction. Journal of agricultural and food chemistry.Journal of Agricultural and Food Chemistry. 2019, 67 (42), 11577-11583. (IF=3.911)

55. Jian Chen* Yang Zhao. Xing-Cong Li. Jin-Hao Zhao*. Pyridine alkaloids in the venom of imported fire ants. Journal of Agricultural and Food Chemistry.  2019, 67, 41, 11388-11395. (IF5 =3.911)

54. Sheng Cai, Nana Shao, Yuanyuan Chen, Anbang Li, Jie Pan, Huajian Zhu, Hongbin Zou, Su Zeng, Lianli Sun,* and Jinhao Zhao*. Enantioselective Reduction of α,β-Unsaturated Ketones and Aryl Ketones by Perakine Reductase. Organic Letters. 2019, 21: 4411-4414  (IF =6.492)

53. Yong Yang, Jinxin Che, Biao Wang,b Yizhe Wu,a Binhui Chen,a Liang Gao,c Xiaowu Dong* and Jinhao Zhao*. Visible-light-mediated guest trapping in a photosensitizing porous coordination network: metal-free C-C bond-forming modification of metal-organic frameworks for aqueous-phase herbicide adsorption.Chemical Communications.2019,55, 5383-5386. (IF =6.290)

52. Yong Yang, Jingli Cheng, Biao Wang, Yirong Guo, Xiaowu Dong, and Jinhao Zhao*. An amino-modified metal-organic framework (type UiO-66-NH2) loaded with Cd(II) and Pb(II) ions for simultaneous electrochemical immunosensing of triazophos and thiacloprid. Microchimica Acta2019186: 101(IF=5.7)

51. Jinhao Zhao, Zhouchen Lin, Shaowei Fang, Xinrui Xie, Huanhuan Wang, Zhenfeng Pang, Jing Zhang, Xueqian Kong, Ming Lei*. Photoexcitation of self-n-doped fullerene ammonium halides: The role of halide ion and a possible synergistic dual-redox cycle mechanism within their aggregate. Journal of Photochemistry & Photobiology A: Chemistry. 373(2019): 131-138 (IF=2.89)

2018

50. 程敬丽肖豆鑫郑敏赵金浩*. S -茚虫威的晶型研究及杀虫活性比较农药学学报2018, 20(3): 294-300.

49. 李中珊,程敬丽,李安邦,赵金浩*,杜永均,朱国念香根草挥发性成分提取分离及其农用生物活性研究进展,农药学学报2018, 203):259-269.

48. Jin-Hao Zhao, Yong Yang, Jin-Xin Che, Jun Zuo, Xiao-Hua Li, Yong-Zhou Hu, Xiao-Wu Dong,* Liang Gao,* Xin-Yuan Liu,* Compartmentalization of Incompatible Polymers within Metal-Organic Framework towards Homogenization of Heterogeneous Hybrid Catalysts for Tandem Reactions. Chemistry - A European Journal. 2018,  24(39) : 9903-9909. (IF=5.16)

47. LikunWang1Jinhao Zhao1, Laura Delgado-Moreno, Jingli Cheng, YichenWang, Sufen Zhang, Qingfu Ye, WeiWang*. Degradation and metabolic profiling for benzene kresoxim-methyl using carbon-14 tracing. Science of the Total Environment. 2018(637-638) 1221-1229. (IF=4.61)

46. Can-Liang Ma, Jin-Hao Zhao(共同一作), Yong Yang, Min-Kui Zhang, Chao Shen, Rong Sheng,Xiao-Wu Dong & Yong-Zhou Hu. A Copper-Catalyzed Tandem Cyclization Reaction of Aminoalkynes with Alkynes for the Construction of Tetrahydropyrrolo[1,2-a]quinolones Scaffold. Scientific Reports, 2017, 7: 16640

45.Ting-TingYao, Dou-XinXiao, Zhong-ShanLi, Jing-Li Cheng, Shao-WeiFang, Yong-Jun Du,Jin-HaoZhao*, Xiao-Wu Dong,* and Guo-NianZhu. Design,Synthesis, Fungicidal Evaluation of Novel Pyrazole-furanand Pyrazole-pyrrole Carboxamide as Succinate Dehydrogen as Inhibitors.Journal of Agricultural and Food Chemistry2017, 65(26), 5397-5403.

44.Ting-Ting Yao,Shao-Wei Fang, Zhong-Shan Li, Dou-Xin Xiao, Jing-Li Cheng, Hua-Zhou Ying, Yong-Jun Du, Jin-Hao Zhao* , Xiao-Wu Dong*Discovery of Novel Succinate Dehydrogenase Inhibitors by the Integration of insilico Library Design and Amide Feature-based Pharmacophore Mapping.Journal of Agricultural and Food Chemistry, 2017, 65(15), 3204–3211.

43. Ting-Ting Yao, Xing-Guo Liu,Jing-Li Cheng, Cheng-Yuan Zhu, Wen-Hu Zhan, Jin-Hao Zhao,Xiao-Wu Dong*. Integration of Pharmacophore Mapping and Molecular Dockingin Sequential Virtual Screening: toward the Discovery of Novel JAK2 Inhibitors. Rsc Advances 2017, 7, 10353-10360.

42. Jinhao Zhao, Likun Wang, Jingli Cheng, Wei Wang,* Qingfu Ye*. Fate Characterization of Benzene Kresoxim-Methyl (a StrobilurinFungicide) in Different Aerobic Soils. Journal of Environmental Quality. 2017.3

41.Jing-Li Cheng , Min Zheng, Ting-Ting Yao ,Xiao-Liang Li , Jin-Hao Zhao*, Min Xia  and Guo-Nian Zhu. Synthesis, antifungal activity and QSAR study of novel trichodermin derivatives. Journal of Asian Natural Products Research. 2015, 17(1): 47-55

40. Ting-Ting Yao, Li-Kun Wang, Jing-Li Cheng, Yong-Zhou Hu, Jin-Hao Zhao* and Guo-Nian Zhu. Optimization of pyrethroid and repellent on fabrics by microencapsulation technique against Aedes albopictus . Medical and veterinary entomology.2015,29 (1): 37-

39. Ting-Ting Yao, Jing-Li Cheng, Bing-Rong Xu, Min-Zhe Zhang, Yong-zhou Hu, Jin-Hao Zhaoa* and Xiao-Wu Dong* . Support Vector Machine (SVM) Classification Model Based Rational Design of Novel Tetronic Acid Derivatives as Potent  Insecticidal and Acaricidal Agents. RSC Advances,2015, 5, 49195-49203.

38. 王丽坤,郑乐贵,程敬丽,赵金浩*,朱国念红火蚁信息素及其在化学防治中的应用研究进展农药学学报2015,175):497-504

37.Min Zheng, Ting-Ting Yao, Xiao-Jun Xu, Jing-Li Cheng, Jin-Hao Zhao*, Guo-Nian Zhu. Synthesis and biological evaluation of novel trichodermin derivatives as antifungal agents. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2014, 24(15): 3565-3568.

36.Jin-Hao Zhao* , Sheng-Hong Lai, Lu-Lu Ruan, Jing-Li Cheng, Cheng-Xia Tan, Guo-Nian Zhu, Structure, bioactivity and implications for environmental remediation of complexes comprising the fungicide hexaconazole bound to copper. Pest Management Science. 2014,70228-233. 

35. Jing-Li Cheng, Xin-Rui He, Zong-Cheng Wang, Jian-Gong Zhang,  Jin-Hao Zhao,*  and Guo-Nian Zhu. Metabolism-based synthesis, biological evaluation and SARs analysis of spirotetramat analogues as potential lipid biosynthesis inhibitors.  Pest Management Science.  201369: 1121–1130

34. JinhaoZhao, XiaojunXu, JingliCheng, YongZhoua, Chulong Zhang, Xiaoming Ou,WeikeSu, and Guonian Zhu, SynthesisandantifungalactivitiesofTrichoderminderivativesasfungicidesonricechemistry & biodiversity. 2013, 10: 600-611.

33.Bing-Rong Xu, Xing-Rui He, Jing-Li Cheng and Jin-Hao Zhao*. 3-(2-Bromo-4-fluoro-phenyl)-acrylic acid 3-(2,5-dimethyl-phenyl)-8-methoxy-2-oxo-1-aza-spiro[4.5]dec-3-en-4-yl ester. Acta Cryst. (2013). E69, o1064-o1065.

32. Xing-Rui He, Bing-Rong Xu, Jing-Li Cheng and Jin-Hao Zhao. (1’S,4’S )-5-(2,5-Dimethylphenyl)-4’-methoxy-6-oxa-3-azaspiro[bicyclo[3.1.0]hexane-2,1’-cyclohexan]-4-one. Acta Cryst (2013). E69, o453

31.徐小军赖生洪,季明华,朱国念,赵金浩*.弥拜霉素类似物的合成、表征和杀虫活性研究.有机化学,,2012,32,1084-1092.

30.JinhaoZhao,JiangongZhang,BingrongXu,ZongchengWang,JingliCheng,GuonianZhu.Design,SynthesisandAnalysisontheQuantitativeStructureActivityRelationshipsof4-PhenylAcylSubstituted3-(2,5-dimethylphenyl)-4-hydroxy-1-azaspiro[4.5]dec-3-ene-2,8-dioneDerivatives. Journal of Agricultural and Food Chemistry, 2012,60:4779-4787

29.Jin-HaoZhao,Zong-ChengWang,Ming-HuaJi,Jing-LiCheng,Guo-NianZhuandChuan-MingYu.Synthesisandbioactivityevaluationofnovelspiromesifenderivatives.PestManagementScience.2012,68(1):10-15TOP SCI

28.J.H.Zhao,Y.L.Zhang,L.W.Wang,J.Y.Wang,C.L.Zhang. Bioactive secondary metabolites from Nigrospora sp LLGLM003, an endophytic fungus of the medicinal plant Moringa oleifera Lam. World Journal of Microbiology & Biotechnology, 2012,28:2107-2112.

27.Jin-HaoZhao,Xiao-JunXu,Ming-HuaJi,Jing-LiCheng,Guo-NianZhu.Design,SynthesisandBiologicalActivitiesofMilbemycinAnalogues.Journal of Agricultural and Food Chemistry,2011,59(6)1453-1469

26.张建功阮璐璐,赵金浩,朱国念. An Unexpected Hydrolysis Productfrom Strobilurin Fungicide: Azoxystrobin.ChineseJ.Struct.Chem.2011,30(8),1132-1136.

25.赵金浩*,王宗成,周勇,朱国念,俞传明.螺环季酮酸衍生物的合成及生物活性研究,有机化学2011,31(10):1631-1638.

24.WANGZong-Cheng,XuBing-Rong,CHENGJing-Li,YUChuan-Ming,ZHAOJin-Hao.SynthesisandCrystalStructureof2-Oxo-3-phenyl-1-oxaspiro[4.5]dec-3-en-4-yl4-chlorobenzoate.ChineseJournalof Structural Chemistry, 2011,30(11):1675-1679.

23.Zong-chengWang. Jing-liCheng. Jin-haoZhao*, FengYu. 3-(tert-butyl)-2-oxo-1-oxaspiro[4.5]dec-3-en-4-yl4-chlorobenzoate.ActaCryst.(2011).E67,o2804.

22.Xiao-JunXu,Xiao-LiangLi,Jing-liCheng,Jin-haoZhao*.4-(E)-3-(2-chlorophenyl)acryloyloxytrichodermin((E)-12,13-epoxytrichethec-9-ene-8-(E)-3-(2-chlorophenyl)acryloyloxyoxime).ActaCryst.(2011). E67, o2834.

21.JinHaoZHAO,MingHuaJIb,XuHuiXU,JingLiCHENG,GuoNianZHU*.Synthesisanaloguesofmilbemycinandtheirbioactivityevaluation.ChineseChemicalLetters,2010,21(11):1391-1394.

20.ZHAOJin-Hao,JIMing-Hua,SUNYa-Quan,CHENGJing-Li,ZHUGuo-Nian.SynthesisandCrystalStructureof2-Methoxy-benzoicacid2-oxo-3-(2,4,6-trimethyl-phenyl)-1-oxa-spiro[4.4]non-3-en-4-ylester.ChineseJournalofStructuralChemistry,2010,29(9):1297-1300.

19.ZHOUYong,XUXu-Hui,CHENGJing-Li,ZHUGuo-Nian,ZHAOJin-Hao*.SynthesisandCrystalStructureofMesitylAceticAcid3-Mesityl-2-oxo-1-oxaspiro[4,4]non-3-en-4-ylEster.ChineseJournalofStructuralChemistry,2010,29(4):517-518.

18.赵金浩,周勇,徐旭辉,朱烈,朱国念,程敬丽.N-(取代噻唑-2-)-菊酰胺类化合物的合成及生物活性研究.有机化学2010,30(5):719-725.

17.Jin-HaoZhao,YongZhou,Jing-LiCheng,Chuan-MingYu,Guo-NianZhu*.3-(2,4-Dichlorophenyl)-2-oxo-1-oxa-spiro[4.5]dec-3-en-4-ylacetate.ActaCryst.(2010).E66,o208.

16.Jin-HaoZhao,YongZhou,Jian-GongZhang,Jing-LiCheng,Fu-ChengLin*.DihalogenatedTrichodermin(4--Acetoxy-9,10-dibromo-12,13-epoxytrichothec).ActaCryst.(2010).E66,o210.

15.Xu-huiXu,Zong-cheng.Wang,Jing-liCheng,YongZhouandJin-haoZhao*Trichodermin(12,13-epoxytrichethec-9-en-4b-yl4-fluorobenzoate)ActaCryst.(2010).E66,o2097.

14.Chuan-mingYu,Zong-chengWang,HuanZhou,Ming-huaJi,Jin-haoZhao*.3-Mesityl-2-oxo-1-oxaspiro[4.4]non-3-en-4-ylbenzoate0.ActaCryst.(2010).E66,o1624

13.JingLiCheng,YongZhou,JinHaoZhao,ChulongZhang,FuChengLin*.SynthesisandantifungalactivityofTrichoderminderivatives.ChineseChemicalLetters,2010,21(09):1037-1040. 12.JinHaoZhao,MingHuaJi,XuHuiXu,JingLiCheng,GuoNianZhu.Syntheticderivativesofspiromesifenandtheirbioactivityresearch.ChineseChemicalLetters,2009,20(11):1307-1310.11.ZHAOJin-hao,ZHOUYong,XUXu-hui,CHENGJing-li,ZHUGuo-nian*.SynthesisandCrystalStructureof3-(2,4-dichlorophenyl)-4-dydroxy-5-cyclohexanyl-Δ3-dihydrofuran-2-one.ChineseJournalofStructuralChemistry,2009,28(7):837-840.

10.Jin-HaoZhao,YongZhou,Guo-nianZhuandJing-LiCheng*4-Hydroxy-3-mesityl-1-oxaspiro[4.4]non-3-en-2-one.ActaCryst.(2009).E65,0755

9.Chuan-MingYu,YongZhou,Jing-LiChengandJin-HaoZhao*.3-Mesityl-2-oxo-1-oxaspiro[4,4]non-3-en-4-yl-2-(4-chlorophenyl)-3-methylbutyrate.ActaCryst.(2009).E65,0183

8.Ming-HuaJi,MinXia,Guo-NianZhuandJin-HaoZhao*.3-Mesityl-2-oxo-1-oxaspiro

[4.4]non-3-en-4-yl4-chlorobenzoateActaCryst.(2009).E65,0705

7.Jing-LiCheng,YongZhou,Fu-ChengLin,Jin-HaoZhao*,Guo-NianZhu.Trichodermol(4a-hydroxy-12,13-epoxytrichothec-9-ene).ActaCryst.(2009).E65,02897

6.YongZhou,Jing-LiCheng,Guo-NianZhu.Jin-HaoZhao*3-(2,4-dichloro-phenyl)-2-oxo-1-oxaspiro[4,5]dec-3-en-4-yl4-chlorobenzoate.ActaCryst.(2009).E65,02992

5.Jing-LiCheng,Jin-HaoZhao,Guo-NianZhuandFu-ChengLin*.2-(4-Chlorophenyl)-3-methyl-N-(5-methylthiazol-2-yl)butanamide.ActaCryst.(2009).E65,0184

4.JinhaoZhao,FengZhao,YanguangWang,HaiboLi,QijunZhang,DanielGuenard,QiufuGe,ErqingWei,HaoJiang,YihangWu,LinWang,HualiangJiang,FranáoiseGueritte,XiumeiWu,ristopherH.K.Cheng,Shoei-ShengLee,andYuZhao*,SynthesisofA/BRingAnalogsofTerritremBandEvaluationofTheirBiologicalActivities,HELVETICACHIMICAACTA.2004,87(7)1832-18

3.JinHaoZHAO,YanGuangWang,HaiBoLI,FengZHAO,LeiXiangYANG,HuaBAI,ShoeiShengLee,YuZHAO*.Synthesisof2-en-1-one-ebelactonylBenzoatesofTerritremBAnaloguesfromJujubogenia.Chinese Chemical Letters200516(1)11-14

2.JinHaoZhao,JingLiCheng,GuonianZhu.2-(4-chlorophenyl)-3-methyl-N-(thiazo-2-yl)butanamide.Acta Cryst.,2006E620840-841

1.FengZHAO,JinHaoZHAO,HaiBoLI,LeiXiangYANG,HuaBAI,YanGuangWang,ShoeiShengLee,YuZHAO*.TwoSerisofSynthesisTerritremBAnaloguesandtheirBiologicalActivities.Chinese Chemical Letters2005,16(4): 457-460

 

已授权发明专利

31. 赵金浩李中珊汪彪王忠燕程敬丽杜永均, 蚜虫天敌瓢虫引诱剂,申请号:201910132778.0,申请日期:2019.02.21 授权日: 2021.06.22

30. Jinhao Zhao, Zhongshan Li, Biao Wang, Zhongyan Wang, Jingli Cheng, Yongjun Du Attractant of Ladybugs, Aphid's Natural EnemyUS 16/851,096 授权日:2021.04.21

29. 赵金浩,赵洋,程敬丽卤代新戊酰基吡喃葡萄糖及其用于SGLT2抑制剂的制备方法. 申请号:201811047732.0. 申请日:2018.09.10,授权日:2021.02.23

28. 赵金浩,姚停停,程敬丽,李中珊,赵洋,董晓武具有杀菌活性的JAK2激酶抑制剂及其虚拟筛选方法,申请号:201710399061.3,申请日:2017.05.31,授权日:2020.11.24 

27. 赵金浩,杨勇,程敬丽,杜永均. 美国白蛾性信息素中间体的合成方法. 专利号:ZL 201810035036.1,申请日:2018.01.15,授权日:2020.08.21  

26. 赵金浩,肖豆鑫,程敬丽,朱国念,李红叶.纳米代森锰锌的制备方法. 申请号:201711490378.4 授权日:2020.04.28

25. 赵金浩,程敬丽,程城,肖豆鑫,李中珊,朱国念. 纳米噻唑锌的制备方法,申请号:201710215759.5 授权日:2019.03.16(专利转让给企业)

24. 程敬丽,程城,赵金浩,肖豆鑫,李中珊,朱国念. 纳米噻唑锌单剂、复配组合物及其用途,申请号:201710225993.6,授权日:2019.03.16专利转让给企业)

23. 赵金浩,姚停停,赵洋,程城程敬丽,朱国念,取代吡唑环类衍生物及用途 ,申请号:201510961071.2,授权日:2018.03.27

22. 程敬丽,赵金浩,郑敏,朱国念精茚虫威的晶型,申请号:201510542484.7,授权日:20180309

21. 赵金浩黄国传程敬丽,赵洋杨勇. (R)-N-叔丁氧羧基联苯丙氨醇的合成方法申请号:201610094826.8,授权日:20171205(专利许可给企业)

20. 陈志远,程敬丽,王丽坤, 赵洋,赵金浩.  2,2-乙基-3,6-二甲基吡嗪的合成方法,申请号: 201510654305.9,授权日:2017.11.21

19. 程敬丽,黄国传,赵金浩,赵洋,杨勇.  (R)-N-叔丁氧羰基联苯丙氨醇的制备方法,申请号:201610095174.X,授权日:2017.05.31

18、程敬丽,赵金浩,郑敏,姜忠义,郑乐贵.农用杀虫剂茚虫威中间体的合成法,申请号:201410453895.4,授权日:2016.08.17

17、程敬丽姚停停黎小亮赵金浩章初龙林福呈.木霉菌素C8不饱和酸酯及其衍生物申请号:201410018923.X,授权日:2016.08.17

16赵金浩,程敬丽,张建功,赖声洪,徐冰融,朱国念.苯基螺环肟醚烯醇酯类化合物及其用途. 201310276124.8, 授权日:2016.04.27

15赵金浩,程敬丽,姜忠义,郑敏,左军农用杀虫剂茚虫威高纯度关键中间体的制备方法,申请号:201410459551.4,授权日:2016.03.30

14、赵洋,赵金浩,程敬丽,郑敏,黎小亮,章初龙,王国平,林福呈木霉菌素C8肟醚类衍生物及其用途申请号:201310482552.6,授权日:2016.01.06

13赵金浩,郑敏,程敬丽,朱国念精茚虫威的晶型及其无定形形式申请号:201310474575.2,授权日:2016.01.20

12赵金浩,王宗成,程敬丽,朱国念苯基螺环酮烯醇酯类化合物及其用途.申请号:201010604623.1,授权日期:2013.1.2

11赵金浩程敬丽,徐旭辉,朱国念. 2-氨基-5--N,3-二甲基苯甲酸胺的制备法.申请号:200910096460.8,授权日:2012.07.25(专利许可6年,15万)

10. 赵金浩,王宗成,程敬丽,朱国念苯基螺环酮烯醇酯类化合物及其用途申请号:201010604623.1 授权日期:2013.01.02

9. 赵金浩程敬丽徐旭辉朱国念. 2-氨基-5--N,3-二甲基苯甲酸胺的制备法申请号:200910096460.8 授权日:2012.07.25

8. 赵金浩王宗成程敬丽朱国念苯基螺环酮烯醇类化合物及其用途申请号:201010538025.9,授权日:2012.07.11

7. 赵金浩徐旭辉程敬丽朱国念具有农药活性的弥拜霉素衍生物及其用途, 申请号:200910097270.8,授权日:2012.07.11

6. 赵金浩程敬丽周勇徐旭辉王国平章初龙林福呈朱国念木霉菌素类衍生物及其防治病原菌的用途.  申请号:201010117859.2. 授权日:2012.02.29 

5. 赵金浩周勇程敬丽徐旭辉朱国念螺螨酯衍生物及其合成方法和用途.申请号:200810060324.9, 授权日 2011.5.4

4. 赵金浩俞海明程敬丽周勇朱国念螺甲螨酯衍生物及其合成方法和用途申请号:200810060325.3, 授权日 2010.11.17

3. 赵金浩戴金贵徐振元一种O,O-二乙基硫代磷酰氯残夜的处理方法申请号:200710070720.5,授权日:2010.6.9

2. 赵金浩徐旭辉周勇程敬丽朱国念一种螺甲螨酯的制备方法,申请号:200810060254.7,授权日 2010.6.16

1. 赵金浩程敬丽,徐旭辉周勇朱国念一种螺螨酯的合成方法  申请号:200810059921.X, 授权日: 2010.6.2